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Docking molecular aplicado ao estudo da formação de complexos entre análogos de resveratrol e derivados de 1,2,3-triazol e a enzima COX-2
(Universidade Federal de São Carlos, 2011-12-14)
Prostaglandin H synthases (PGHS), or cyclooxygenases (COX), are known to exist in at least two isoforms, COX-1 and COX-2, encoded by different genes. COX s play a central role in the inflammatory cascade by converting ...
Nanopartículas de grafite para carreamento de antiinflamatórios não esteroidais por estudos de docking molecular
(Universidade Federal de São Carlos, 2013-08-13)
The non steroidal anti-inflammatory drugs have been known for over 100 years and has been widely used by mankind. However cause adverse effects, since gastrointestinal complications to cardiac diseases many of these symptoms ...