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Síntese e caracterização de Complexos de Pd(II) com potencial atividade citotóxica e inibidores das enzimas Topoisomerase II
(Universidade Federal de São Carlos, 2018-05-29)
It is known that cancer is a set of more than 100 diseases which are the second largest cause of death in the world. There are several factors related to the growth of tumors, showing different pathway for the planning of ...
Citotoxicidade de complexos de rutênio contendo aminoácidos sulfurados em células tumorais
(Universidade Federal de São Carlos, 2016-07-28)
The work presents the synthesis and characterization of three new ruthenium II complexes containing sulfur amino acids, to evaluate the probable influence of the amino acids on the complexes cytotoxic activity. The complexes ...
Complexos fosfínicos de rutênio contendo o ligante 2,2’-dipiridilamina: síntese, caracterização e avaliação de suas atividades citotóxicas e de interação com DNA
(Universidade Federal de São Carlos, 2016-02-29)
This work aims the synthesis, characterization and evaluation of the biological activities of a series of mixed ligand ruthenium (II) phosphine complexes the containing 2,2’-dipyridylamine ligand. Furthermore, the studies ...
Tetra(tien-2-il)porfirina e seus complexos com metais da primeira-série de transição: síntese, caracterização, investigação da citotoxicidade e interação com DNA
(Universidade Federal de São Carlos, 2020-07-21)
Cancer is a generic term for over 100 diseases with uncontrolled cell growth. Each year, all cancer forms are responsible for millions of deaths worldwide and are the leading cause of deaths linked to disease. Therefore, ...
Síntese e caracterização de complexos de Prata (I): investigação da citotoxidade e interação com o DNA
(Universidade Federal de São Carlos, 2020-06-23)
The inorganic compound, cisplatin, is used on a large scale to different types of cancer. This complex acts in DNA structure by covalent bonds. However, the chemotherapy agent presents several side effects and some tumors ...
Citotoxidade e mecanismo de ação de complexos Ru(II)/2-mercapto-4(3H)quinazolinona em células de câncer de pele
(Universidade Federal de São Carlos, 2023-02-28)
Ruthenium biphosphynic complexes combined with mercapto ligands have shown low IC50 values and good selectivity indexes (SI) in different tumor lines studied, which has motivated the development of ruthenium compounds with ...